SYN-1030-M001
SYN-1030-M005
SYN-1030-M010
SYN-1030-M050
102991-478EA
74.77
USD
InStock
102991-478
102991-480
102991-482
102991-484
Canertinib ≥95%
Canertinib
Canertinib is an orally bio-available EGFR inhibitor with potential anti-neoplastic and radio-sensitizing activities. It has IC(50) values of 1.5nM and 9.0nM against EGFR and ErbB2 respectively, with no activity against PDGFR, FGFR, InsR, PKC, or CDK1/2/4.